| Bioactivity | GPR17 modulator-1 (Compound 2-046) is a modulator for G protein-coupled receptor 17 GPR17, with an IC50<10 nM for hGPR17 in CHO. GPR17 modulator-1 exhibits moderate pharmacokinetic characteristics in mice. GPR17 modulator-1 ix blood-brain barrier (BBB) permeable[1]. |
| CAS | 3039853-91-0 |
| Formula | C15H12ClF3N4O4S |
| Molar Mass | 436.79 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Han X, et al., Gpr17 modulators and uses thereof. WO2024104462. |