Bioactivity | GPR132 antagonist 1 (GPR132-B-160, Compound 25) is a GPR132 antagonist with an EC50 value of 0.075 μM. GPR132 antagonist 1 has promote insulin secretion activity with an EC50 value of 0.7 μM[1]. |
Target | EC50: 0.075 μM (GPR132); 0.7 μM (insulin secretion activity). |
Name | GPR132 antagonist 1 |
CAS | 898211-21-7 |
Formula | C18H17NO5S |
Molar Mass | 359.40 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. 焦宁, 等. Gpcr调节剂及其应用. 专利. CN116903563A. |