Bioactivity | GPR119 agonist 3 (Compound 21b) is an orally active agonist of GPR119 with an EC50 value of 3.8 nM for hGPR119. Additionally, GPR119 agonist 3 exhibits hypoglycemic effects and can be used in research on type 2 diabetes and obesity[1]. |
Target | EC50: 3.8 nM (hGPR119). |
CAS | 2097502-14-0 |
Formula | C30H40N4O3 |
Molar Mass | 504.66 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. La H, et al. Discovery of 1, 4-Disubstituted Cyclohexene Analogues as Selective GPR119 Agonists for the Treatment of Type 2 Diabetes[J]. Journal of Medicinal Chemistry, 2025. |