Bioactivity | GPR109 receptor agonist-2 (Compound 5) is a selective GPR109a agonist with a pEC50 of 5.53[1]. | ||||||||||||
Target | pEC50: 5.53 (GPR109a) | ||||||||||||
Name | GPR109 receptor agonist-2 | ||||||||||||
CAS | 957129-38-3 | ||||||||||||
Formula | C7H10N2O2 | ||||||||||||
Molar Mass | 154.17 | ||||||||||||
Appearance | 固体 | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
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Reference | [1]. Skinner PJ, et al. Fluorinated pyrazole acids are agonists of the high affinity niacin receptor GPR109a. Bioorg Med Chem Lett. 2007 Oct 15;17(20):5620-3. |