| Bioactivity | GLP-1R modulator C5 is an allosteric modulator enhancing GLP-1 binding to GLP-1R via a transmembrane site (EC50 1.59 ± 0.53 μM). | ||||||||||||
| Name | GLP-1R modulator C5 | ||||||||||||
| CAS | 421578-93-0 | ||||||||||||
| Formula | C24H21NO3 | ||||||||||||
| Molar Mass | 371.43 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
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| Reference | [1]. Wang J, et al. Allosteric Modulators Enhancing GLP-1 Binding to GLP-1R via a Transmembrane Site. ACS Chem Biol. 2021 Nov 19;16(11):2444-2452. |