Bioactivity | GLP-1R modulator C16 is an allosteric modulator enhancing GLP-1 binding to GLP-1R via a transmembrane site (EC50 8.43 ± 3.82 μM). | ||||||||||||
Name | GLP-1R modulator C16 | ||||||||||||
CAS | 875005-43-9 | ||||||||||||
Formula | C21H26ClFN2O3 | ||||||||||||
Molar Mass | 408.89 | ||||||||||||
Appearance | Solid | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
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Reference | [1]. Wang J, et al. Allosteric Modulators Enhancing GLP-1 Binding to GLP-1R via a Transmembrane Site. ACS Chem Biol. 2021 Nov 19;16(11):2444-2452. |