| Bioactivity | GID4 Ligand 3 (compound 16) is a binder of GID4 with an Kd value of 110 μM in vitro and an IC50 value of 148.5 μM. GID4 Ligand 3 can be used for the research related to cereblon and Von Hippel-Lindau[1]. |
| Target | IC50: 148.5 μM (GID4) |
| Invitro | GID4 Ligand 3 (0-1000 μM; 30 min) binds with GID4 with a Kd value of 110 μM[1]. |
| Name | GID4 Ligand 3 |
| CAS | 340007-39-8 |
| Formula | C10H12N2OS |
| Molar Mass | 208.28 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Chana CK, et al. Discovery and Structural Characterization of Small Molecule Binders of the Human CTLH E3 Ligase Subunit GID4. J Med Chem. 2022 Sep 18. |