Bioactivity | FR260010 free base is a selective 5-HT2C receptor antagonist, with a Ki value of 1.1 nM[1]. |
Target | Ki: 1.1 nM (5-HT2C receptor). |
Name | FR260010 free base |
CAS | 374555-75-6 |
Formula | C22H19N5 |
Molar Mass | 353.42 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Katsuya Harada, et al. Activation of the serotonin 5-HT2C receptor is involved in the enhanced anxiety in rats after single-prolonged stress. Pharmacol Biochem Behav. 2008 Mar;89(1):11-6. |