| Bioactivity | FGFR4-IN-1 is a potent inhibiotr of FGFR4 with IC50 of 0.7 nM. | ||||||||||||
| Invitro | FGFR4-IN-1 significantly inhibits the proliferation of HuH-7 hepatocellular carcinoma cells with IC50 of 7.8 nM[1]. | ||||||||||||
| Name | FGFR4-IN-1 | ||||||||||||
| CAS | 1708971-72-5 | ||||||||||||
| Formula | C24H27N7O5 | ||||||||||||
| Molar Mass | 493.52 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
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| Reference | [1]. Ring-fused bicyclic pyridyl derivatives as fgfr4 inhibitors. WO 2015059668 A1? |