Bioactivity | FAP-IN-1 is a fibroblast activation protein (FAP) inhibitor with an IC50 value of 3.3 nM. FAP-IN-1 can be used for the research of cancer[1]. |
Target | IC50: 3.3 nM (FAP). |
Name | FAP-IN-1 |
Formula | C65H88F2N12O18 |
Molar Mass | 1363.46 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Wang Y, et al. High Affinity and FAP-Targeted Radiotracers: A Potential Design Strategy to Improve the Pharmacokinetics and Tumor Uptake for FAP Inhibitors. J Med Chem. 2023 Jul 13;66(13):8614-8627. |