| Bioactivity | Eplerenone (Epoxymexrenone) is a selective, highly specific and orally active aldosterone blocker (SAB). Eplerenone also is a selective mineralocorticoid receptor antagonist (MRA) with IC50 value of 0.081 μM. Eplerenone can be used for the research of hypertension, atherosclerosis, chronic systolic heart failure (HF) and cardiovascular (CV)[1][2]. | ||||||||||||
| Invitro | Eplerenone inhibits the human mineralocorticoid receptor with IC50 value of 0.081 μM[2]. | ||||||||||||
| Name | Eplerenone | ||||||||||||
| CAS | 107724-20-9 | ||||||||||||
| Formula | C24H30O6 | ||||||||||||
| Molar Mass | 414.49 | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
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