Bioactivity | Endothelial lipase inhibitor-1 is a potent endothelial lipase inhibitor with an IC50 of 49 nM. | ||||||||||||
Target | IC50: 49 nM (Endothelial lipase) | ||||||||||||
Name | Endothelial lipase inhibitor-1 | ||||||||||||
CAS | 1466427-02-0 | ||||||||||||
Formula | C22H22N4O4 | ||||||||||||
Molar Mass | 406.43 | ||||||||||||
Appearance | Solid | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
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Reference | [1]. Hu CH, et al. Discovery and synthesis of tetrahydropyrimidinedione-4-carboxamides as endothelial lipase inhibitors. Bioorg Med Chem Lett. 2018 Dec 15;28(23-24):3721-3725. |