| Bioactivity | EZH2-IN-22 (example 92) is a potent EZH2 inhibitor with IC50 values of <0.00051, <0.00051, 0.00052 µM for EZH2 (Y641N), EZH2 (Y641F), EZH2 (wt), respectively. EZH2-IN-22 shows antiproliferation activity[1]. |
| CAS | 2766231-05-2 |
| Formula | C36H50N4O8 |
| Molar Mass | 666.80 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Wei Peng, et al. Polysubstituted benzene compound and preparation method and use thereof. French.WO2020020374A1. |