| Bioactivity | EST64454 (compound 9k) 是一种选择性具有口服活性的 sigma-1 受体拮抗剂，Ki 为 22 nM。EST64454 可用于疼痛的研究。 |
| CAS | 1351438-26-0 |
| Formula | C18H22F2N4O2 |
| Molar Mass | 364.39 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Yeste S, et al. Preliminary in Vitro Assessment of the Potential of EST64454, a Sigma-1 Receptor Antagonist, for Pharmacokinetic Drug-Drug Interactions. Biol Pharm Bull. 2020;43(1):68-76. |