Bioactivity | ERK2-IN-4 (Compound 6o) is an effective and selective ERK2 inhibitor with a Ki of 0.006 μM. ERK2-IN-4 inhibits the ERK signaling pathway and can be used in cancer research[1]. |
CAS | 933786-58-4 |
Formula | C22H17Cl2FN4O2 |
Molar Mass | 459.30 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Aronov, Alex M et al. “Flipped out: structure-guided design of selective pyrazolylpyrrole ERK inhibitors.” Journal of medicinal chemistry vol. 50,6 (2007): 1280-7. |