| Bioactivity | ERK2-IN-3 (compound 2) is a inhibitor of ERK2, and inhibits Erk2WT and Erk2DS1 activation loop phosphorylation, with IC50 of 5 μM and 42 nM, respectively[1]. |
| Target | 5 μM and 42 nM（Erk2WT and Erk2DS1 ）. |
| Name | ERK2-IN-3 |
| CAS | 1415050-57-5 |
| Formula | C26H21F3N4O |
| Molar Mass | 462.47 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Hari SB, et al. Conformation-selective ATP-competitive inhibitors control regulatory interactions and noncatalytic functions of mitogen-activated protein kinases. Chem Biol. 2014;21(5):628-635. |
ERK2-IN-3
CAS: 1415050-57-5 F: C26H21F3N4O W: 462.47
ERK2-IN-3 (compound 2) is a inhibitor of ERK2, and inhibits Erk2WT and Erk2DS1 activation loop phosphorylation, with IC5
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