| Bioactivity | EPZ0025654 (GSK3536023) is an inhibitor for protein arginine methyltransferases 4 (PRMT4) (which is also known as coactivator associated arginine methyltransferase 1 CARM1), with IC50 of 3 nM[1]. |
| CAS | 1888328-89-9 |
| Formula | C29H33ClN8O3 |
| Molar Mass | 577.08 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Li ASM, et al., Chemical probes for protein arginine methyltransferases. Methods. 2020 Mar 15;175:30-43. |