| Bioactivity | EP4 receptor antagonist 4 is an EP4 receptor agonist with the human pEC50 value of 6.3[1]. |
| Invitro | EP4 receptor antagonist 4 (24 h) treatment shows agonism in HEK293 cells stably transfected with hEP4[1].EP4 receptor antagonist 4 (30 min) treatment shows agonism (pEC50<5) and antagonism (pIC50<5)[1]. Cell Viability Assay[1] Cell Line: |
| Name | EP4 receptor antagonist 4 |
| CAS | 691869-12-2 |
| Formula | C19H14N2OS |
| Molar Mass | 318.39 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Joannes Theodorus Maria Linders, et al. Bicyclic derivatives as ep4 agonists. WO2008092860A1 |