| Bioactivity | EP300/CBP-IN-1 (compound 172) is a potent EP300/CBP inhibitor with IC50s of 2.3 nM and 2.1 nM for CBP BRD and EP300 BRD, respectively. EP300/CBP-IN-1 has the inhibitory effect on the proliferation of prostate cancer CWR22RV1 cells[1]. |
| Name | EP300/CBP-IN-1 |
| CAS | 2638507-71-6 |
| Formula | C30H32ClFN4O4 |
| Molar Mass | 567.05 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Lei Fan, et al. An EP300/CBP inhibitor. CN112574189A. |
EP300/CBP-IN-1
CAS: 2638507-71-6 F: C30H32ClFN4O4 W: 567.05
EP300/CBP-IN-1 (compound 172) is a potent EP300/CBP inhibitor with IC50s of 2.3 nM and 2.1 nM for CBP BRD and EP300 BRD,
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