| Bioactivity | EP1-antagonist-1 is a EP1 antagonist with a pKi of 7.54 and an pIC50 of 8.5[1]. |
| Target | pIC50: 8.5 (EP1)pKi: 7.54 (EP1) |
| Name | EP1-antagonist-1 |
| CAS | 851204-35-8 |
| Formula | C19H15BrCl2N2O3 |
| Molar Mass | 470.14 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. McKeown SC, et al. Identification of novel pyrazole acid antagonists for the EP1 receptor. Bioorg Med Chem Lett. 2006 Sep 15;16(18):4767-71. Epub 2006 Jul 14. |