| Bioactivity | ELA-21 (human) is an apelin receptor agonist with a pKi of 8.52. ELA-21 (human) completely inhibits Forskolin-induced cAMP production and stimulates β-arrestin recruitment with subnanomolar potencies. ELA-21 (human) is an agonist in G-protein-dependent and -independent pathways[1]. |
| Name | ELA-21 (human) |
| CAS | 2245073-05-4 |
| Sequence | Leu-Arg-Lys-His-Asn-Cys-Leu-Gln-Arg-Arg-Cys-Met-Pro-Leu-His-Ser-Arg-Val-Pro-Phe-Pro (Disulfide bridge: Cys6-Cys11) |
| Shortening | LRKHNCLQRRCMPLHSRVPFP (Disulfide bridge: Cys6-Cys11) |
| Formula | C112H184N40O25S3 |
| Molar Mass | 2587.14 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
ELA-21 (human)
CAS: 2245073-05-4 F: C112H184N40O25S3 W: 2587.14
ELA-21 (human) is an apelin receptor agonist with a pKi of 8.52. ELA-21 (human) completely inhibits Forskolin-induced cA
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