| Bioactivity | E2508 is an orally active corticotropin-releasing factor 1 receptor antagonist with a Ki value of 11 nM for hCRF1[1]. |
| CAS | 685886-34-4 |
| Formula | C36H47N3O7S |
| Molar Mass | 665.84 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Takahashi Y, et al. Synthesis and structure-activity relationships of pyrazolo[1,5-a]pyridine derivatives: potent and orally active antagonists of corticotropin-releasing factor 1 receptor. J Med Chem. 2012 Jun 14;55(11):5255-69. |