| Bioactivity | Dyrk1A-IN-11 (compound 166) is a potent dual-specificity tyrosine phosphorylation- regulated 1A (DYRK1A) inhibitor with an EC50 value of 0.0021 µM. Dyrk1A-IN-11 inhibits the Phospho-Tau (Thr212) with an EC50 value of 0.0361 µM[1]. |
| CAS | 3058626-26-6 |
| Formula | C23H23F5N8O |
| Molar Mass | 522.47 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Gopi Kumar Mittapalli, et al. Pyrrolo[2,1-f][1,2,4]triazines and preparation and uses thereof. French, WO2024211797A1. |
Dyrk1A-IN-11
CAS: 3058626-26-6 F: C23H23F5N8O W: 522.47
Dyrk1A-IN-11 (compound 166) is a potent dual-specificity tyrosine phosphorylation- regulated 1A (DYRK1A) inhibitor with
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