| Bioactivity | Dynorphin A TFA is an endogenous opioid peptide involved in inhibitory neurotransmission in the central nervous system (CNS). Dynorphin A TFA is a highy potent kappa opioid receptor (KOR) agonist, and is also an agonist for other opioid receptors, such as mu (MOR) and delta (DOR). Dynorphin A TFA can induce neuronal death, and can be used in the research of neurological disease[1][2]. |
| Invitro | Dynorphin A TFA (10 μM, 4 h/72 h) increases caspase-3 activity and the level of cytochrome c released from mitochondria in mouse striatal neurons, and induces neuronal death[3].dynorphin A TFA (33 μM, 4 h) elevates [Ca2+]i and causes a significant loss of neurons[4].dynorphin A TFA (1 μM) inhibits the release of vasopressin (VP) from the isolated neural lobe[5]. Cell Viability Assay[3] Cell Line: |
| Name | Dynorphin A TFA |
| Formula | C101H156F3N31O25 |
| Molar Mass | 2261.50 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Dynorphin A TFA
CAS: F: C101H156F3N31O25 W: 2261.50
Dynorphin A TFA is an endogenous opioid peptide involved in inhibitory neurotransmission in the central nervous system (
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