| Bioactivity | DSP-2230 is a selective Nav1.7/Nav1.8 blocker[1][2]. | ||||||||||||
| Target | Nav1.7/Nav1.8 | ||||||||||||
| Name | DSP-2230 | ||||||||||||
| CAS | 1233231-30-5 | ||||||||||||
| Formula | C20H20F3N5O2 | ||||||||||||
| Molar Mass | 419.40 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
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| Reference | [1]. Bagal SK, et al. Voltage gated sodium channels as drug discovery targets. Channels (Austin). 2015;9(6):360-6. [2]. Sara Sabina Hadida-Ruah, et al. Sulfonamides as modulators of sodium channels. |