| Bioactivity | DS43260857 is a potentNaV1.7inhibitor, which has a high inhibitory effect on both human and mouse NaV1.7. The IC50 values of DS43260857 for hNaV1.1, hNaV1.5, hNaV1.7, mNaV1.7 are 6.6, 14, 0.015 and 0.061 μM, respectively[1]. |
| Target | IC50:6.6μM(hNaV1.1),14μM(hNaV1.5), 0.015μM(mNaV1.7),0.061μM(mNaV1.7) |
| Name | DS43260857 |
| CAS | 1612158-07-2 |
| Formula | C19H16F3N3O3S |
| Molar Mass | 423.41 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Narayan Karanjule, et al. N-Aryl Indoles as a Novel Class of Potent NaV1.7 Inhibitors. ACS Med Chem Lett. 2023 May 24;14(6):788-793. |
DS43260857
CAS: 1612158-07-2 F: C19H16F3N3O3S W: 423.41
DS43260857 is a potentNaV1.7inhibitor, which has a high inhibitory effect on both human and mouse NaV1.7. The IC50 value
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