| Bioactivity | Cruzain-IN-1 is a covalent and reversible Cruzain inhibitor, with an IC50 of 10 nM. | ||||||||||||
| Name | Cruzain-IN-1 | ||||||||||||
| CAS | 1199523-24-4 | ||||||||||||
| Formula | C14H10F2N6 | ||||||||||||
| Molar Mass | 300.27 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
|
||||||||||||
| Reference | [1]. Lee GM, et al. Mapping inhibitor binding modes on an active cysteine protease via nuclear magnetic resonance spectroscopy. Biochemistry. 2012 Dec 18;51(50):10087-98. |