PeptideDB

Crinecerfont

CAS: 752253-39-7 F: C27H28ClFN2OS W: 483.04

Crinecerfont (SSR-125543) hydrochloride is a potent, orally active, non-peptide CRF1 receptor antagonist. Crinecerfont c
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This product is for research use only, not for human use. We do not sell to patients.

Bioactivity Crinecerfont (SSR-125543) hydrochloride is a potent, orally active, non-peptide CRF1 receptor antagonist. Crinecerfont can be used for Classic congenital adrenal hyperplasia (CAH) research[1].
Target IC50: CRF1 receptor
Name Crinecerfont
CAS 752253-39-7
Formula C27H28ClFN2OS
Molar Mass 483.04
Transport Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Reference [1]. Global Safety and Efficacy Registration Study of Crinecerfont for Congenital Adrenal Hyperplasia (CAHtalyst).