PeptideDB

Crinecerfont hydrochloride

CAS: 321839-75-2 F: C27H29Cl2FN2OS W: 519.50

Crinecerfont (SSR-125543) hydrochloride is a potent, orally active, non-peptide CRF1 receptor antagonist. Crinecerfont c
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This product is for research use only, not for human use. We do not sell to patients.

Bioactivity Crinecerfont (SSR-125543) hydrochloride is a potent, orally active, non-peptide CRF1 receptor antagonist. Crinecerfont can be used for Classic congenital adrenal hyperplasia (CAH) research[1].
Target IC50: CRF1 receptor
Name Crinecerfont hydrochloride
CAS 321839-75-2
Formula C27H29Cl2FN2OS
Molar Mass 519.50
Appearance Solid
Transport Room temperature in continental US; may vary elsewhere.
Storage

4°C, sealed storage, away from moisture and light

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)

Reference [1]. Global Safety and Efficacy Registration Study of Crinecerfont for Congenital Adrenal Hyperplasia (CAHtalyst).