Cloxacepride

CAS: 65569-29-1 F: C22H27Cl2N3O4 W: 468.37

Cloxacepride is an orally active and potent antiallergic agent. Cloxacepride is a CaM (calmodulin) antagonist. Cloxacepr

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Bioactivity	Cloxacepride is an orally active and potent antiallergic agent. Cloxacepride is a CaM (calmodulin) antagonist. Cloxacepride has anti-PCA (passive cutaneous anaphylaxis) activity[1][2].
In Vivo	Cloxacepride 的口服 ED50 值为 46-49 mg/kg，与茶碱 (Theophylline, HY-B0809) 和静脉注射 2 mg/kg 色甘酸二钠 (DSCG) 后立即激发相当[1]。在抗原攻击前 15 或 60 分钟口服给药时，Cloxacepride 具有抗 PCA 活性[1]。 MCE has not independently confirmed the accuracy of these methods. They are for reference only.
CAS	65569-29-1
Formula	C22H27Cl2N3O4
Molar Mass	468.37
Transport	Room temperature in continental US; may vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Reference	[1]. Metz G, et al. Cloxacepride and related compounds: a new series of orally active antiallergic compounds. J Med Chem. 1983 Jul;26(7):1065-70.

Dimethyl succinate

C.I. Direct violet 66