| Bioactivity | ChemR23-IN-1 (compound 2) is a ChemR23 inhibitor with IC50s of 38 nM and 100 nM for human and mouse ChemR23, respectively. ChemR23-IN-1 inhibits chemotaxis of CAL-1 triggered by Chemerin in vitro[1]. |
| Target | IC50: 38 nM (human ChemR23 ) and 100 nM (mouse ChemR23) |
| Name | ChemR23-IN-1 |
| CAS | 2378640-10-7 |
| Formula | C28H29N7O2 |
| Molar Mass | 495.58 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Takamichi Imaizumi, et al. The design, synthesis and evaluation of 2-aminobenzoxazole analogues as potent and orally efficacious ChemR23 inhibitors. Bioorg Med Chem. 2020 Sep 1;28(17):115622. |
ChemR23-IN-1
CAS: 2378640-10-7 F: C28H29N7O2 W: 495.58
ChemR23-IN-1 (compound 2) is a ChemR23 inhibitor with IC50s of 38 nM and 100 nM for human and mouse ChemR23, respectivel
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