Bioactivity | Cenupatide (UPARANT) is a Urokinase-type plasminogen activator receptor (uPAR) inhibitor. Cenupatide has anti-angiogenic and anti-inflammatory efficacy[1]. |
Name | Cenupatide |
CAS | 1006388-38-0 |
Sequence | Ac-Arg-{Aib}-Arg-{aMePhe}-NH2 |
Shortening | Ac-R-{Aib}-R-{aMePhe}-NH2 |
Formula | C28H47N11O5 |
Molar Mass | 617.74 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Filippo Locri, et al. UPARANT is an effective antiangiogenic agent in a mouse model of rubeosis iridis. J Mol Med (Berl). 2019, 97, 9. [2]. Cai Yuan, et al. Development of inhibitors for uPAR: blocking the interaction of uPAR with its partners. Drug Discov Today. 2021, 26, 4. |