| Bioactivity | Cavα2δ-IN-1 shows high selectivity for voltage-gated calcium channels Cavα2δ-1 (Ki 6 nM) versus Cavα2δ-2 (Ki ＞ 10000 nM). |
| Name | Cavα2δ-IN-1 |
| CAS | 2416957-09-8 |
| Formula | C18H27N5O |
| Molar Mass | 329.44 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Fernández A, et al. Piperazinyl Bicyclic Derivatives as Selective Ligands of the α2δ-1 Subunit of Voltage-Gated Calcium Channels. ACS Med Chem Lett. 2021 Oct 5;12(11):1802-1809. |