| Bioactivity | Cathepsin K inhibitor 4 is a potent carbohydrazide Cathepsin K inhibitor with IC50s of 13 nM, 269 nM, 296 nM for human, rat, mouse Cathepsin K, respectively[1]. |
| Target | IC50: 13 nM (Cathepsin K), 38 nM (Cathepsin B), 8.9 nM (Cathepsin L), 792 nM (Cathepsin S) and 3.2 nM (Cathepsin F) |
| Name | Cathepsin K inhibitor 4 |
| Sequence | Boc-Phe-Leu-{NHNH-CO-NHNH}-Leu-{Z} |
| Shortening | Boc-FL-{NHNH-CO-NHNH}-L-{Z} |
| Formula | C35H51N7O8 |
| Molar Mass | 697.82 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Sylvie Desmarais, et al. Pharmacological inhibitors to identify roles of cathepsin K in cell-based studies: a comparison of available tools. Biol Chem. 2009 Sep;390(9):941-8. |
Cathepsin K inhibitor 4
CAS: F: C35H51N7O8 W: 697.82
Cathepsin K inhibitor 4 is a potent carbohydrazide Cathepsin K inhibitor with IC50s of 13 nM, 269 nM, 296 nM for human,
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