Bioactivity | CaMKK2-IN-1 is a selective, ligand-efficient inhibitor of CaMKK2, with IC50 of 7 nM[1]. |
Target | CaMKK2 (IC50 = 7 nM) |
Name | CaMKK2-IN-1 |
Formula | C22H22N2O3 |
Molar Mass | 362.42 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Young Chen, et al. Identification of Small Molecule Inhibitors and Ligand Directed Degraders of Calcium/Calmodulin Dependent Protein Kinase Kinase 1 and 2 (CaMKK1/2). J Med Chem. 2023 Dec 14;66(23):15750-15760. |