| Bioactivity | CV1808 (2-Phenylaminoadenosine) is a non-selective A2 adenosine receptor (A2 AR) agonist with Kis of 76 and 1450 nM for A2A and A3 adenosine receptor subtypes, respectively[1]. | |||||||||
| Invitro | CV1808 demonstrates an inhibitory effect on anti-IgE-induced activation at 100 μM[1].In the presence of Forskolin (1 μM in PC12 cells; 10 μM in Jurkat cells) the EC50 value for CV1808 is 2 μM[2]. | |||||||||
| Name | CV1808 | |||||||||
| CAS | 53296-10-9 | |||||||||
| Formula | C16H18N6O4 | |||||||||
| Molar Mass | 358.35 | |||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | |||||||||
| Storage |
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