PeptideDB

CK-963

CAS: 2851991-63-2 F: C27H36N6O5S W: 556.68

CK-963 is an activator for cardiac troponin (cTnC) with Ki of 11.5 μM. CK-963 exhibits activity in enhancing cardiac co
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Bioactivity CK-963 is an activator for cardiac troponin (cTnC) with Ki of 11.5 μM. CK-963 exhibits activity in enhancing cardiac contractility in Sprague-Dawley rats[1].
Target Ki: 11.5 μM (cTnC)
In Vivo CK-963 (0.5 mg/kg,静脉注射) 在 SD 大鼠体内的药代动力学分析显示,其在肝脏血液中的清除率 Route
CAS 2851991-63-2
Formula C27H36N6O5S
Molar Mass 556.68
Transport Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Reference [1]. Collibee SE, et al., Cardiac Troponin Activator CK-963 Increases Cardiac Contractility in Rats. J Med Chem. 2024 Mar 7.