Bioactivity | CK-963 is an activator for cardiac troponin (cTnC) with Ki of 11.5 μM. CK-963 exhibits activity in enhancing cardiac contractility in Sprague-Dawley rats[1]. |
Target | Ki: 11.5 μM (cTnC) |
In Vivo | CK-963 (0.5 mg/kg,静脉注射) 在 SD 大鼠体内的药代动力学分析显示,其在肝脏血液中的清除率 Route |
CAS | 2851991-63-2 |
Formula | C27H36N6O5S |
Molar Mass | 556.68 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Collibee SE, et al., Cardiac Troponin Activator CK-963 Increases Cardiac Contractility in Rats. J Med Chem. 2024 Mar 7. |