| Bioactivity | CHIR-2279 is a high-affinity ligand (Ki=5 nM) for the α1-adrenergic receptor and can be further studied as a drug lead compound[1]. |
| CAS | 158198-45-9 |
| Formula | C34H36N4O4 |
| Molar Mass | 564.67 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Zuckermann, et al. Discovery of nanomolar ligands for 7-transmembrane G-protein-coupled receptors from a diverse N-(substituted) glycine peptoid library. Journal of medicinal chemistry 37.17 (1994): 2678-2685. |