Bioactivity | CGI 560 is an inhibitor for Bruton's tyrosine kinase (BTK) with an IC50 of 400 nM. |
Target | IC50: 400 nM (Bruton's tyrosine kinase) |
CAS | 845269-74-1 |
Formula | C29H27N5O |
Molar Mass | 461.56 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Lv J, et al., Development of Bruton's Tyrosine Kinase Inhibitors for Rheumatoid Arthritis. Curr Med Chem. 2018;25(42):5847-5859. |