| Bioactivity | CEP1347-VHL-02 is a PROTAC targeting MLK3. CEP1347-VHL-02 consists of PROTAC target protein ligand CEP-1347 (HY-10412), E3 ubiquitin ligase ligand (S,R,S)-AHPC-Me (HY-112078) and PROTAC Linker Amino-PEG3-CH2COOH (HY-140189), of which the target protein ligand activity control is CEP-1347-acid (HY-168027), and the conjugate of E3 ubiquitin ligase ligand + Linker is (S,R,S)-AHPC-Me-CO-CH2-PEG3-NH2 (HY-131387)[1]. |
| Target | MLK3 |
| Formula | C61H72N8O11S3 |
| Molar Mass | 1189.47 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |