CBP/p300-IN-21_product_DataBase

CAS: 1065581-69-2 F: C19H16ClNO4 W: 357.79

CBP/p300-IN-21 (Compound 5d) is a selective CBP/p300 inhibitor (IC50: 0.07 and 1.755 μM for p300 and CBP). CBP/p300-IN-

This product is for research use only, not for human use. We do not sell to patients.

Bioactivity	CBP/p300-IN-21 (Compound 5d) is a selective CBP/p300 inhibitor (IC50: 0.07 and 1.755 μM for p300 and CBP). CBP/p300-IN-21 decreases H3K18Ac level. CBP/p300-IN-21 inhibits growth of 4T1 tumor growth in mice[1].
Target	0.07 and 1.755 μM for p300 and CBP
Name	CBP/p300-IN-21
CAS	1065581-69-2
Formula	C19H16ClNO4
Molar Mass	357.79
Transport	Room temperature in continental US; may vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Reference	[1]. Zhong X, et al. Discovery of berberine analogs as potent and highly selective p300/CBP HAT inhibitors. Bioorg Chem. 2023 Sep;138:106597.

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