| Bioactivity | CB2 receptor antagonist 3 (compound (S)-1) is an inverse agonist of the cannabinoid receptor CB2R with Kd=39 nM. CB2 receptor antagonist 3 can be used as a tool to synthesize a variety of CB2R probes[1]. |
| Target | Kd: 39 nM (CB2R) |
| Name | CB2 receptor antagonist 3 |
| Formula | C33H46N4O2 |
| Molar Mass | 530.74 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Carreira E et al. Flipping the GPCR Switch: Structure–Based Development of Selective Cannabinoid Receptor 2 Inverse Agonists[J]. 2023. |
CB2 receptor antagonist 3
CAS: F: C33H46N4O2 W: 530.74
CB2 receptor antagonist 3 (compound (S)-1) is an inverse agonist of the cannabinoid receptor CB2R with Kd=39 nM. CB2 rec
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