Bioactivity | CB2 PET Radioligand 1 (compound [18F]9) is a PET Radioligand targeting to hCB2 (Ki=7.7 nM). CB2 PET Radioligand 1 is prepared with Cu-mediated 18F-fluorination. CB2 PET Radioligand 1 shows high brain uptake in a murine model of neuroinflammation[1]. |
Target | Ki: 7.7 nM (human CB2) |
In Vivo | CB2 PET Radioligand 1 (compound [18F]9) |
Name | CB2 PET Radioligand 1 |
Formula | C20H19F3N4O |
Molar Mass | 388.39 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Kallinen A, et al. Synthesis and Preclinical Evaluation of Fluorinated 5-Azaindoles as CB2 PET Radioligands. ACS Chem Neurosci. 2023 Aug 16;14(16):2902-2921. |