Bioactivity | Bz-Dab(NBD)-AwFpP-Nle-NH2 (Compound 5B) is a potent fluorescent antagonist of NK2 receptor, with a pKi of 8.87 nM (Ex=340 nm, Em=505 nm)[1]. |
CAS | 161238-74-0 |
Sequence | Bz-{Dab(NBD)}-Ala-{d-Trp}-Phe-{d-Pro}-Pro-{Nle}-NH2 |
Shortening | Bz-{Dab(NBD)}-A-{d-Trp}-F-{d-Pro}-P-{Nle}-NH2 |
Formula | C56H65N13O11 |
Molar Mass | 1096.20 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Bradshaw CG, et al. Synthesis and characterization of selective fluorescent ligands for the neurokinin NK2 receptor. J Med Chem. 1994 Jun 24;37(13):1991-5. |