Blue FPG-A trisodium

CAS: 78617-94-4 F: C29H17ClN7Na3O11S3 W: 840.10

Blue FPG-A trisodium is a selective antagonist of P2X1 receptor and P2Y1 receptor with IC50 values of 35.5 μM and 2.6

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Bioactivity	Blue FPG-A trisodium is a selective antagonist of P2X1 receptor and P2Y1 receptor with IC50 values of 35.5 μM and 2.6 μM, respectively. Blue FPG-A trisodium is a structural isomer of the components of Reactive Blue 2 (RB2)[1].
Invitro	Blue FPG-A trisodium (RB 2 para) (1-100 μM) 抑制 α、β-亚甲基 ATP (α、β-MeATP) 诱导的大鼠输精管 (RVD) 收缩和 5’-o-(2-硫代二磷酸腺苷) (ADPβS) 诱导的卡巴胆碱 (Carbachol，HY-B1208) 预处理的豚鼠结肠带 (GPTC) 的松弛[1]。
Name	Blue FPG-A trisodium
CAS	78617-94-4
Formula	C29H17ClN7Na3O11S3
Molar Mass	840.10
Transport	Room temperature in continental US; may vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Reference	[1]. Glänzel M, et al. Constitutional isomers of Reactive Blue 2 - selective P2Y-receptor antagonists? Eur J Med Chem. 2003 Mar;38(3):303-12.