Bioactivity | BM30 is a selective peptidomimetic NTMT1 and NTMT2 inhibitor (IC50: 0.89 μM for NTMT1)[1]. |
CAS | 2606862-05-7 |
Sequence | {4-Hydroxyphenylacetyl}-Pro-Lys-Arg-NH2 |
Shortening | {4-Hydroxyphenylacetyl}-PKR-NH2 |
Formula | C25H40N8O5 |
Molar Mass | 532.64 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Mackie BD, et al. Selective Peptidomimetic Inhibitors of NTMT1/2: Rational Design, Synthesis, Characterization, and Crystallographic Studies. J Med Chem. 2020 Sep 10;63(17):9512-9522. |