| Bioactivity | Benzarone (Fragivix) is a potent human uric acid transporter 1 (hURAT1) inhibitor, with an IC50 of 2.8 μM in oocyte. Benzarone could lower uric acid serum levels[1]. | ||||||||||||
| Target | IC50: 2.8 μM (hURAT1 in oocyte) | ||||||||||||
| Name | Benzarone | ||||||||||||
| CAS | 1477-19-6 | ||||||||||||
| Formula | C17H14O3 | ||||||||||||
| Molar Mass | 266.30 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
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| Reference | [1]. Wempe MF, et, al. Developing potent human uric acid transporter 1 (hURAT1) inhibitors. J Med Chem. 2011 Apr 28;54(8):2701-13. |