| Bioactivity | Beloxepin (Org 4428) is an orally active synaptosomal noradrenalin reuptake inhibitor and a 5-HT2 receptor antagonist. Beloxepin shows about 100-fold less affine for other monoamine carriers. Beloxepin has antidepressant and pain-relieving effects[1][2]. |
| CAS | 135928-30-2 |
| Formula | C19H21NO2 |
| Molar Mass | 295.38 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Lorenzo Di Cesare Mannelli, et al. α2 Adrenoceptor: a Target for Neuropathic Pain Treatment. Mini Rev Med Chem. 2017;17(2):95-107. [2]. Craig T Hartrick. Noradrenergic reuptake inhibition in the treatment of pain. Expert Opin Investig Drugs. 2012 Dec;21(12):1827-34. |