Bioactivity | BRD4 Inhibitor-29 (SQ-17) is a BRD4 inhibitor, with an IC50 of <100 nM. BRD4 Inhibitor-29 shows antiproliferative effect against prostate cancer cells[1]. |
Name | BRD4 Inhibitor-29 |
CAS | 902563-50-2 |
Formula | C21H28N2O3 |
Molar Mass | 356.46 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Haiyang Zhong, et al. Discovery of Novel Inhibitors of BRD4 for Treating Prostate Cancer: A Comprehensive Case Study for Considering Water Networks in Virtual Screening and Drug Design. J Med Chem. 2024 Jan 11;67(1):138-151. |