Bioactivity | BQ-3020 (TFA) is a selective agonist of ETB receptor, inhibits [125I]ET-1 binding to ETB receptor with an IC50 of 0.2 nM in cerebellum, and causes vasoconstriction[1]. | ||||||
Name | BQ-3020 TFA | ||||||
Sequence | N-Acetyl-Leu-Met-Asp-Lys-Glu-Ala-Val-Tyr-Phe-Ala-His-Leu-Asp-Ile-Ile-Trp | ||||||
Shortening | N-Acetyl-LMDKEAVYFAHLDIIW | ||||||
Formula | C98H141F3N20O27S | ||||||
Molar Mass | 2120.35 | ||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||
Storage | Sealed storage, away from moisture and light
*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light) |